Mumasumbu akawanda, kusanganisira moyo, pamwe nemariti, itsvo, airways nemamwe matukisi, pane beta-adrenergic receptors. Izvo zvinokonzera zvakanyanya, uye dzimwe nguva zvinotyisa, kuzviita kwemuviri kunodarika uye kudzvinyirira ("hit kana kumhanya"). Kuti kuderedze basa ravo mukurapa, beta-blockers inoshandiswa - urongwa hwemishonga kubva kune iri boka rezvemasikirini rakakura zvikuru, rinobvumira kusarudza mishonga yakakodzera kwazvo kune mumwe murwere mumwe nomumwe.
Non-selective beta-blockers
Kune marudzi maviri eAdrenoreceptors - beta-1 uye beta-2. Apo kushandiswa kokutanga kwakavharwa, zvinotevera mamiriro emwoyo zvinowanikwa:
- kuderedza mumoyo wehuwandu uye nguva zhinji;
- kuderedza kuwedzera kweropa;
- kudzvinyirirwa kwekunyengedza mwoyo.
Kana iwe ukavhara beta-2-adrenoreceptors, pane kuwedzera kweropa kumirisana yemidziyo yeropa nezwi:
- chibereko (muvakadzi vane pamuviri);
- bronchi;
- arterioles.
Kugadzirira kubva muboka re nonselective beta-blockers kuita zvisarudzo, kuderedza basa rezvinhu zvose zviripo.
Mishonga inotevera inoreva mishonga iri kuongororwa:
- Oxprenolol;
- Propranolol;
- Pindolol;
- Anaprilin;
- Sotalol;
- Penbutolol;
- Nadolol;
- Timolol;
- Inderal;
- Obsidan;
- Bopindolol;
- Okupres-E;
- Sandinorm;
- Levobunolol;
- Wistagen;
- Korgard;
- Obinol;
- Wistagan;
- Oxprenolol;
- Tracicore;
- Koretal;
- Vickin;
- Sotalol;
- Timolol;
- Viskaldix;
- Sotagexal;
- Okumol;
- Sotaleks;
- Arutimol;
- Xalacom;
- Okumed;
- Fotil nevamwe.
Sarudza beta-blockers
Kana mushonga wacho uchishanda sarudzo uye unoderedza kushanda kwe beta-1-adrenergic receptors, iyo inosarudzwa. Zvakakosha kuziva kuti madhiragi akadaro anonyanya kufanirwa mune kurapwa kwemararamiro emwoyo, kunze kwekuti, anounza mashoma emigumisiro.
Rwendo rwezvinodhaka kubva muboka re cardioselective beta-blockers rwechizvarwa chitsva:
- Betacard;
- Atenolol;
- Tenolol;
- Prinorm;
- Bisoprolol;
- Tenoric;
- Hypoten;
- Bisocardium;
- Tenoretik;
- Bisogamma;
- Concor;
- Lokren;
- Coronale;
- Betaxolol;
- Metoprolol;
- Betoptik;
- Corvitol;
- Vasocardine;
- Logimax;
- Egilok;
- Metocard;
- Amzok;
- Kwete-tiketi;
- Esmolol;
- Breviblock;
- Nebivolol;
- Talinolol;
- Cordanum;
- Acebutolol.
Zvakaipa zvinokonzerwa ne beta-blockers
Zvinhu zvisina kunaka zvinowanzokonzera kusasarudzwa kwemishonga. Izvi zvinosanganisira zvinhu zvinotevera:
- bradycardia ;
- zviratidzo zvemoyo kusakatika;
- arterial hypotension;
- kurwadziwa mubhokisi;
- kurara kunetseka kana kusuruvara;
- chizoro;
- kukanganwa kwepfungwa uye kukwanisa kuisa pfungwa;
- kuora mwoyo;
- maonero ekuona uye anoongorora;
- kushanda kwakadzika;
- kusafarira;
- headaches;
- nausea;
- akaoma muromo;
- kuvhara kana kubatwa;
- kurutsa;
- kurwadziwa mu epigastrium uye mumatumbo;
- manyore kusangana;
- bronchospasm;
- dyspnea;
- kunetseka kufema;
- aplastic anemia;
- thrombocytopenic purpura;
- thromboses;
- hypothyroidism;
- kuderedza libido uye potency;
- gynecomastia;
- misuli spasms;
- arthralgia ;
- kudengenyeka;
- myasthenia gravis;
- kuoma kwemukoko mucosa;
- kuonekwa kusakanganisika;
- kuderera kwehuwandu hwemvura yakasunungurwa yakabudiswa;
- conjunctivitis;
- kunhuwa kweganda;
- urticaria;
- kutuka kukuru;
- kunzwisisika kweganda kune ultraviolet;
- peremia ye epidermis;
- kudzokazve kweporioriasis;
- alopecia (reversible);
- kurwadziwa mushure.
Kazhinji, mushure mekudzivisa adrenoblocker, kune "kubvisa chirwere" muchimiro chekuwedzera kwakasimba uye kusingagumi kweropa, nguva dzakawanda dze angina pectoris.