Nonsteroidal anti-inflammatory drug in the modern pharmaceutical market is presented in a variety of forms - both in powders, and in tablets, and in injections, and, of course, in the form of ointments and gels. Chimwe cheNSAID dzinonyanya kufarirwa nenzira yejeri inogona kudanwa Diclofenac. Izvi zvinokonzerwa nezvikonzero zvakasiyana-siyana: kutanga, mishonga haina mari yakakwirira, uye yechipiri, inoshanda chaizvo, uye, chechitatu, mukurumbira kwezita remishonga inotsigirwa nemamwe maitiro - majekiseni akafanana uye mahwendefa.
Kugadzirwa kweGel Diclofenac
Diclofenac kubudirira anomiririra kupesana-kupisa kwete steroid agents uye ine gel kubva ku diclofenac sodium.
Izvo zvinhu zvinobatsira zvinobatsira gel kupinda zviri nani kuva maviri uye kuchengetedza zvinhu zvavo kwenguva refu ndeizvi:
- ethanol yakagadziriswa;
- propylene glycol;
- triethanolamine;
- mutambi;
- methyl lauryl hydroxybenzonate;
- lavender oil;
- mvura yakachena.
Kubudiswa kusununguka uye kuiswa kwemajeri Diclofenac
Gel Diclofenac inowanikwa mualuminium tubes ye 50 uye 40 g.
Mukuwedzera kumhepo, kuiswa kwezvinhu zvakasiyanawo:
- Diclofenac gel 5% - pa 1 g yehutano inokwana 50 mg ye diclofenac sodium;
- Diclofenac gel 3% - 1 g ye gel account ye 30 mg ye diclofenac sodium;
- Diclofenac gel 1% - 1 g ye gel is 10 mg yeganda rinoshandiswa - diclofenac sodium.
Diclofenac marashi haachipo, chete gel inowanikwa.
Pharmacological properties ye gel Diclofenac
Diclofenac iyi mishonga inobata marwadzo, uyewo inonzi anti-inflammatory properties. Inhibisa ma enzymes COX-2 uye COX-1, uye inokanganisawo kuyanana kwe arachidonic acid uye metabolism ye prostaglandin, iyo inoumba chine chekuvhiringidza. Nokudaro, gel rinoderedza kupararira kwekuputika, uye rinodzivirirawo kukura kwarwo mumatunhu akakomberedzwa.
Pamusana pezvinhu izvi, Diclofenac inoshandiswa sekuti decongestant kana kupfugama kunokonzerwa nokuputika. Inorayirwawo kuti chirwere chinorwadza seanesesthetic yepanyika kana kurwadziwa kunokonzerwa nekuputira.
Diclofenac inoderedza kuzvimba mumamiriro ekubatana kwekubatana, kubvisa kuoma. Uyewo munzvimbo dzekuvhiringidza, iye anogona kubvisa marwadzo, kana kunyanya kuderedza.
Diclofenac gel mirayiridzo
Mirayiridzo yekushandiswa kweDiclofenac Gel 5%, uyewo 3% uye 1% haisi yakasiyana. Misiyano iri muhutano hwezvinhu zvinoshanda, uye chinangwa chayo chinoenderana nekuoma kwezviratidzo. Semuenzaniso, Diclofenac gel rine mazamu e5% anoshandiswa kurwara kurwadziwa kwakanyanya mu rheumatism .
Zviratidzo zvekushandisa gel Diclofenac
Diclofenac inorayirwa kune zvirwere zvinotevera:
- rheumatic pathologies - bursitis , tendovaginitis, etc ;;
- Uturu hwepachiviri pamucheto we rheumatism kana kukuvadza kumisungo yemasumbu;
- kuvhiringidzika kwekupedzisira kwemasangano.
Diclofenac gel rinoshandiswa kunze, uye nhamba yekushandiswa kumwe chete kunobva paukuru hwenzvimbo inorwadza.
Zvisinei, pane mazano akawanda ekuti kushandiswa kwegelisi yakasiyana-siyana:
- Diclofenac gel 1% - kushandiswa kumwe chete - kusvika 4 g;
- Diclofenac gel 3% - kushandiswa kumwe chete - kusvika 3 g;
- Diclofenac gel 5% - kushandiswa kamwe chete kusvika 2 g.
Vana vaduku vanopfuura makore gumi nemaviri uye vakuru vanokurudzirwa kushandisa gel 3-4 kazuva nekushanda kwekudzivirira chiedza.
Contraindications kushandiswa kweGel Diclofenac
Diclofenac haigoni kushandiswa mumamiriro ezvinhu anotevera:
- pamuviri (kukurudzirwa 3 trimester);
- lactation;
- vana vezera (kusvika kumakore 6);
- maronda, anopisa;
- zvinokonzera kugadzikana kana chirwere chinokonzerwa nekushandiswa kwemasina asingatori steroidal anti-inflammatory drugs.
Kana pane chirwere chekubuda ropa, Diclofenac Gel 5% inofanira kushandiswa nekuchenjerera.