Antiemetic drug for chemotherapy

Antiemetic zvinodhaka mushure mekemotherapy yakagadzirirwa kuderedza emesis panguva yekugamuchirwa kune varwere vane cytotoxic zvinodhaka. Nyaya yemishonga iyi haigone kushandiswa pasina antiemetic zvinodhaka. Zvichienderana nerudzi rwe cytostatics, marudzi akasiyana-siyana okurutsa anokura, somuenzaniso wakaoma kana kuti anononoka. Yokutanga inowanikwa musi wekutanga mushure mekutanga kurapwa, uye wechipiri-kubva kuchipiri kusvika kunechishanu.

Uyezve munyaya iyo iwe uchaona mazita uye tsanangudzo dzezvinonyanyozivikanwa zvekare zvinonzi antiemetic chemotherapy.

Lorazepam

Icho chinotyisa, chimiro chepoda yakachena, iyo isinganyunyuki mumvura. Chirwere ichi chinoshandiswa zvakanyanya, pakati pezviratidzo hachisi kungorutsa chete, asiwo zvepfungwa, pamwe nezvimwe zvinetso:

Contraindicated kune varwere vane hypersensitivity kune mishonga kana zvikamu zvayo, pamwe chete nevanhu vanotambura-yakavharwa-angle glaucoma, kunyanya kudhakwa uye kudzvinyirira mabasa epakati yenheyo. Izvo hazvikurudzirwi kutora mishonga kuvarwere vane hutachiwana husina simba.

Vakaberekwa uye vakadzi vane pamuviri vane mikana mukushandiswa kwemishonga inonzi Laurazepam, iyo inoti: inorambidzwa zvachose kutora mishonga mumutambo wekutanga wekuita pamuviri, uye munguva yemishonga inorayirwa kurega kunwisa.

Lorazepam ine migumisiro inogona kuitika mu:

Mune zvimwe zviitiko, kuora mwoyo kunogona kuitika. Saka, tora mishonga yacho zvakanyatsokodzera maererano nechiremba wechiremba uye inofanira kunyatsotevera mirairo.

Nezvizhinji zvinopesana nemigumisiro, zvinodhaka zvinonzi Lorazepam zvinoshandiswa kubudirira sechirwere chinopesana neusea mu chemotherapy.

Dronabinol

Dronabinol inowanika mumakutu e 2.5 mg, 5 mg uye 10 mg. Chirwere chacho chinoshandiswa zvakasiyana-siyana-kubva kubatsiro mukurwisa kuora kwemazivi munyaya yeAIDS, kusvika pakurapwa kwekutsvaira nekutuka. Dronabinol inofanira kutorwa katatu pazuva pazuva 5 mg. Nguva yenguva yekurapa inorayirwa nachiremba. Mushonga wacho hauna kukodzera zvakakwana nedoro uye zvinyararire, saka zvakakosha kudzivisa kushandisa kwavo panguva yekurapa naDronabinol.

Mishonga ine mimwe migumisiro yakaipa:

Dronabinol inofanira kutorwa chete sezvinorayirwa nachiremba uye pasi pekutarisirwa kwake.

Pakati pezvinyorwa zvinokonzerwa ne hypersensitivity, zvinetso zvepfungwa, makumbo uye lactation. Vagadziri vanocherechedza kuti kushandiswa kwechirwere muhutachiwana hahuna kudzidza, saka hazvikurudzirwi kuti uzvishandise kune vanaamai vari mberi.

Prochlorperazine

Mishonga iyi ndeyeboka revana, saka rinoshandiswa kurapa varwere vane schizophrenia nemamwe psychoses ane zviratidzo zvehutachiona, asthenia, kusava nehanya uye stuporosis, uye semishonga inorwisa-emeemiti yekunyunyuta shure kwechemotherapy.

Mushonga unofanirwa kutorwa nemuromo mushure mekudya. Pazuva rokutanga rokubvumirwa, unofanira kutora 12.5 - 25 mg uye zuva rega rega, zvishoma nezvishoma uwedzere muyero pamwe chete. Apo zuva nezuva iyo mikoko ichasvika 150 - 300 mg, iwe unoda kumira, uye mumurayi uyu mishonga inotorwa kusvikira pakuguma kwechikoro, iyo inowanzotora mwedzi miviri kusvika mitatu.

Kushandiswa kwehuwandu hwechirwere kunogona kukonzera kubudirira:

Kurwara kwenguva yakareba kunokonzera granulocytopenia.